Aromasin – Exemestane 25mg

ACTIVE HALF-LIFE: 9 HOURS
CLASSIFICATION: STEROIDAL AROMATASE INHIBITOR
DOSAGE: 12.5-25 MG/DAY
ACNE: NO
WATER RETENTION: NO
HBR: NO
HEPATOXITY: NO
AROMATIZATION: NO

Exemestane is a newly developed and powerful anti-estrogen drug that works by hindering the transformation of certain substances in the body into estrogen. It is primarily used in the treatment of breast cancer in post-menopausal women when other treatments have failed. Exemestane specifically targets the enzymes that generate estrogen in various parts of the body of post-menopausal women, which are different from the ovaries in pre-menopausal women. The bodybuilding community has adopted Exemestane for its effectiveness in preventing estrogen conversion that can occur with many steroids.

Many anabolic and androgenic steroids convert into estrogen within the body, which can lead to unwanted effects in men such as gynecomastia, increased fat deposits, and water retention that can obscure muscle definition. Exemestane may help reduce body fat, boost testosterone levels by as much as 60%, and enhance somatomedin, a compound with anabolic properties. Despite its ability to elevate testosterone, Exemestane is generally not used in post-cycle therapy and is most beneficial during a full cycle.

In the bodybuilding realm, the suggested daily dose to prevent estrogen build-up varies from 12.5 mg to 25 mg. Known as one of the most effective anti-estrogen drugs available, Exemestane has been shown to lower estrogen levels by up to 85% in some studies involving women. Dosages can vary significantly depending on individual biology, the strength of steroids, and their dosage. Some may notice tangible results with just 2.5 mg of Exemestane, while others might find that 12.5 mg every other day is sufficient. Selecting the correct dosage is essential, particularly because of the strength of this anti-estrogen, as inadequate estrogen levels could impede muscle development and lower libido.

In men, Exemestane could increase the likelihood of cardiovascular issues. Those who are concerned about heart health might want to explore other anti-estrogen options. Women taking Exemestane for medical reasons might experience a range of side effects, including hot flashes, stomach discomfort, bone health problems, elevated blood pressure, and potential birth defects during pregnancy. As a steroidal suicide aromatase inhibitor, some effects of Exemestane's reduction of estrogen can be long-lasting due to its irreversible binding to estrogen-converting enzymes.

Exemestane is typically available in tablet form, containing around 25 mg of the drug, and can be found in most pharmacies, both in the US and worldwide, under that name.

Keep Exemestane away from children. It is intended for adult use only.